GPCR Solutions
Comprehensive HTRF cellular platform
Cell surface receptor studies and functional assays.
GPCR investigation is among the top priorities in drug discovery research.
Cisbio has supported this area for many years by bringing regularly cutting edge assays and technologies fitted for receptor characterization and for compounds screening and lead optimization
Cisbio expands its offers for functional readouts (second messenger accumulation assays: cyclic-AMP & IP-One) with Cellul'erk, a new assay which allows detection of phosphorylated ERK directly in cells.
The new Tag-lite™ cell-surface receptor platform means Cisbio Bioassays now provides reagents and technology to address the latest evolution in the GPCR drug discovery field.
Features:- Single technology and cellular platform for all GPCR assays
- Unique non-radioactive ligand binding assays
- Miniaturization down to < 10µl
GPCR functional assays
| Second messenger accumulation kits | ||
|---|---|---|
| Gi/Gs | ||
| Gq | ||
| Phosphorylated ERK1/2 detection | ||
| GI/s/q | ||







