GPCR Solutions

Comprehensive HTRF cellular platform


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GPCR cell lines
Cell surface receptor studies and functional assays.

GPCR investigation is among the top priorities in drug discovery research.

Cisbio Bioassays has supported this area for many years by bringing regularly cutting edge assays and technologies fitted for receptor characterization and for compounds screening and lead optimization

Cisbio Bioassays expands its offers for functional readouts (second messenger accumulation assays: cyclic-AMP & IP-One) with Cellul'erk, a new assay which allows detection of phosphorylated ERK directly in cells, and GPCR internalization assay a new service.

Features:
  • Single technology and cellular platform for all GPCR assays
  • Unique non-radioactive ligand binding assays
  • Miniaturization down to < 10µl

GPCR functional assays

Second messengers accumulation kits
Gi/Gs
Gq
Phosphorylated ERK1/2 detection
GI/s/q